SCHEMBL6205006

SCHEMBL6205006

CCCN(CO)c1nc(NCc2ccccc2)c2c(n1)N(C(C)C)NN2C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 9/20 0.44
CDK5 Q00535 6/20 0.44
CDK2 P24941 10/20 0.41
CCNE1 P24864 8/20 0.41
CCNE2 O96020 7/20 0.41
PDE5A O76074 3/20 0.37
PDE4D Q08499 3/20 0.37
PDE6C P51160 2/20 0.37
CCNA2 P20248 2/20 0.37
CCNA1 P78396 1/20 0.37
CCNB1 P14635 2/20 0.36
CDK7 P50613 2/20 0.35
CDK9 P50750 2/20 0.35
CCNT1 O60563 1/20 0.35
CCNH P51946 1/20 0.35
MNAT1 P51948 1/20 0.35
CDK5R1 Q15078 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CSNK1D P48730 1/20 0.35
CLK2 P49760 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204543 0.87 CCNE1 (0.37) CDK1CDK5CDK2CCNE1CCNE2
SCHEMBL6205415 0.87 CDK1 (0.34) CDK1CDK5CDK2CCNE1CCNE2
SCHEMBL6205631 0.86 CCNE2 (0.44) CDK1CDK5CDK2CCNE1CCNE2
SCHEMBL6201113 0.83 CDK1 (0.46) CDK1CDK5CDK2CCNE1CCNE2
SCHEMBL6203902 0.82 CCNE2 (0.31) CDK2CCNE1CCNE2
SCHEMBL6204991 0.81 PKM (0.42) CDK2CCNE1CCNE2CDK9CCNT1
SCHEMBL6204186 0.80 PDE5A (0.36) CDK1CDK5CDK2CCNE1CCNE2
SCHEMBL6204092 0.80 CCNT1 (0.31) CDK5CDK2CCNE1CDK7CDK9
SCHEMBL6206198 0.78 CCNE2 (0.46) CDK1CDK2CCNE1CCNE2
SCHEMBL6203776 0.77 CDK5 (0.46) CDK1CDK5CDK2CCNE1CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed