SCHEMBL6205054

SCHEMBL6205054

O=[N+]([O-])c1c[c]ccc1CBr

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 3/20 0.35
TDP1 Q9NUW8 6/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALOX15 P16050 2/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
CYP3A4 P08684 1/20 0.32
SNCA P37840 1/20 0.32
GPR35 Q9HC97 1/20 0.31
ALOX12 P18054 1/20 0.31
NPC1 O15118 1/20 0.31
RECQL P46063 1/20 0.31
RAB9A P51151 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456636 0.83 PDK1 (0.41) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL3604296 0.81 ALDH1A1 (0.39) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL11152901 0.81 ALDH1A1 (0.56) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL16950649 0.80 MAPT (0.36) ALDH1A1HPGDTSHRTDP1MAPT
SCHEMBL8177420 0.80 POLB (0.39) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL28355811 0.78 ALOX15 (0.40) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL11151232 0.77 ALDH1A1 (0.39) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL28277263 0.77 POLB (0.36) ALDH1A1HPGDTSHRTDP1MEN1
SCHEMBL27420001 0.77 ALDH1A1 (0.40) ALDH1A1HPGDTDP1POLBMAPT
SCHEMBL8876153 0.76 CYP1A2 (0.40) ALDH1A1MEN1KMT2APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1545523-A1 3-&-grave;(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES ASP38 MAP KINASE INHIBITORS Astex Technology Limited (GB) 2005-06-29 EP disclosed
WO-2005002673-A1 RAF KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed
WO-2004004720-A1 3-`(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES AS P38 MAP KINASE INHIBITORS ASTEX TECHNOLOGY LIMITED (GB) 2004-01-15 WO disclosed