SCHEMBL6205608

SCHEMBL6205608

CCCN(CO)c1nc(NCc2cccc(OC(C)=O)c2)c2[nH]nnc2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
STAT3 P40763 2/20 0.36
PDE4D Q08499 2/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
ACHE P22303 3/20 0.33
PDE5A O76074 1/20 0.33
PDE6C P51160 1/20 0.33
MAPT P10636 1/20 0.33
PRUNE1 Q86TP1 1/20 0.32
LMNA P02545 1/20 0.32
SLC26A6 Q9BXS9 1/20 0.32
AURKA O14965 2/20 0.32
RPS6KB1 P23443 2/20 0.32
AURKB Q96GD4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205602 0.87 PARP1 (0.37) PARP1PDE4DHTTSMN1; SMN2PDE4A
SCHEMBL6205328 0.84 PARP1 (0.36) PARP1STAT3PDE4DHTTSMN1; SMN2
SCHEMBL6202760 0.84 CDK1 (0.40) PDE4DSMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL3445270 0.78 CDK1 (0.46) STAT3SMN1; SMN2LMNAAURKA
SCHEMBL6203171 0.77 CCNE1 (0.37) AURKA
SCHEMBL3445690 0.77 STAT3 (0.41) PARP1STAT3HTTSMN1; SMN2MAPT
SCHEMBL3446443 0.76 CDK1 (0.45) PARP1STAT3HTTSMN1; SMN2MAPT
SCHEMBL3445494 0.76 STAT3 (0.40) PARP1STAT3HTTSMN1; SMN2ACHE
SCHEMBL6203495 0.75 PRUNE1 (0.35) PDE4DPDE5APDE6CPRUNE1
SCHEMBL3444313 0.74 CDK1 (0.52) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed