SCHEMBL6205353

SCHEMBL6205353

CN(C)CCNCc1ccc(C=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.45
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
CYP2A6 P11509 2/20 0.42
CYP2A13 Q16696 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
HDAC1 Q13547 1/20 0.41
EPHX2 P34913 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
ALDH1A1 P00352 2/20 0.40
ALDH3A1 P30838 1/20 0.40
ALDH1A3 P47895 1/20 0.40
TERT O14746 1/20 0.40
CHRM2 P08172 1/20 0.38
HRH3 Q9Y5N1 2/20 0.38
BRAF P15056 1/20 0.38
TBK1 Q9UHD2 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10054980 0.87 SIGMAR1 (0.50) OPRM1OPRK1SIGMAR1HDAC1TERT
SCHEMBL13102974 0.79 CHRM2 (0.60) OPRM1OPRK1SIGMAR1HDAC1TERT
SCHEMBL10535689 0.78 CHRM2 (0.58) SIGMAR1ALDH1A1CHRM2TMEM97CA12
SCHEMBL30119829 0.78 KEAP1 (0.49) OPRM1OPRK1SIGMAR1HDAC1TERT
SCHEMBL16268751 0.78 CHRM2 (0.58) EPHX2ALDH1A1CHRM2CA12CA1
SCHEMBL18434706 0.78 CYP2C9 (0.63) OPRM1OPRK1SIGMAR1HDAC1TERT
SCHEMBL3879539 0.78 CHEK1 (0.48) OPRM1OPRK1SIGMAR1HDAC1ALDH1A1
SCHEMBL3037243 0.78 TAAR1 (0.57) OPRM1OPRK1SIGMAR1HDAC1TERT
SCHEMBL18434292 0.78 CARM1 (0.48) OPRM1OPRK1SIGMAR1HDAC1TERT
SCHEMBL133622 0.77 MEN1 (0.64) SIGMAR1HDAC1CHRM2TMEM97MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551841-A1 PYRAZOLOPYRIMIDINES AS KINASE INHIBITORS SmithKline Beecham Corporation (US) 2005-07-13 EP disclosed
WO-2004009602-A1 PYRAZOLOPYRIMIDINES AS KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-01-29 WO disclosed