SCHEMBL6206418

SCHEMBL6206418

COc1cccc2c(=O)c(C(=O)NCc3ccc(CN4CCCCC4)cc3)c[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.60
ALDH1A1 P00352 4/20 0.60
POLB P06746 2/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
NPC1 O15118 1/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
RAB9A P51151 1/20 0.60
MAPK10 P53779 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
HSD17B10 Q99714 1/20 0.60
KDM4E B2RXH2 1/20 0.53
CNR2 P34972 1/20 0.52
CHRM3 P20309 1/20 0.47
HRH3 Q9Y5N1 2/20 0.47
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203895 0.91 POLB (0.49) HPGDALDH1A1POLBMEN1KMT2A
SCHEMBL6206617 0.90 POLB (0.50) HPGDALDH1A1POLBMEN1KMT2A
SCHEMBL6208399 0.85 RAB9A (0.58) HPGDALDH1A1RAB9AHRH3TSHR
SCHEMBL6204183 0.84 POLB (0.72) HPGDALDH1A1POLBMEN1KMT2A
SCHEMBL6206415 0.80 KDM4E (0.60) HPGDALDH1A1POLBHSD17B10KDM4E
SCHEMBL6205208 0.79 CHRM3 (0.53) HPGDALDH1A1POLBMEN1KMT2A
SCHEMBL6205610 0.78 HPGD (0.47) HPGDALDH1A1POLBMEN1KMT2A
SCHEMBL6206035 0.77 MAPT (0.58) HPGDALDH1A1POLBKMT2ANPC1
SCHEMBL6206009 0.77 HPGD (0.58) HPGDALDH1A1POLBNPC1RAB9A
Hydrochloric Acid SCHEMBL6205334 0.76 MAPT (0.57) HPGDALDH1A1POLBKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed