SCHEMBL6206680

SCHEMBL6206680

COc1cccc(-c2cccc(C(=O)O)c2-c2cccc(OC)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 3/20 0.55
PRKAB2 O43741 1/20 0.53
PRKAG1 P54619 1/20 0.53
PRKAA2 P54646 1/20 0.53
PRKAA1 Q13131 1/20 0.53
PRKAG3 Q9UGI9 1/20 0.53
PRKAG2 Q9UGJ0 1/20 0.53
PRKAB1 Q9Y478 1/20 0.53
KDM4E B2RXH2 2/20 0.52
GAA P10253 1/20 0.52
DHODH Q02127 3/20 0.51
AKR1C3 P42330 2/20 0.50
AKR1C2 P52895 2/20 0.50
EDNRB P24530 1/20 0.50
EDNRA P25101 1/20 0.50
RAB9A P51151 1/20 0.49
LMNA P02545 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5085746 0.88 HNF4A (0.63) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL496484 0.88 KDM4E (0.62) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL7796258 0.85 GPR35 (0.55) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL18377850 0.84 AKR1C3 (0.55) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL8202718 0.81 PRKAB2 (0.55) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL27501023 0.80 GPR35 (0.56) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL8887143 0.80 GAA (0.59) KDM4EGAALMNAALDH1A1HPGD
SCHEMBL10471506 0.78 GPR35 (0.55) GPR35PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL1515816 0.78 GAA (0.62) KDM4EGAARAB9ALMNAALDH1A1
SCHEMBL27913989 0.77 WDR5 (0.58) GPR35PRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1503997-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-02-09 EP disclosed
WO-2003097617-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2003-11-27 WO disclosed