SCHEMBL6206683

SCHEMBL6206683

CCC(NC(=O)[CH]C1CCCCC1)C(O)c1nc2ccccc2o1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.44
HDAC3 O15379 7/20 0.39
HDAC4 P56524 7/20 0.39
HDAC1 Q13547 7/20 0.39
HDAC7 Q8WUI4 7/20 0.39
HDAC2 Q92769 7/20 0.39
HDAC10 Q969S8 7/20 0.39
HDAC11 Q96DB2 7/20 0.39
HDAC8 Q9BY41 7/20 0.39
HDAC6 Q9UBN7 7/20 0.39
HDAC9 Q9UKV0 7/20 0.39
HDAC5 Q9UQL6 7/20 0.39
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
CTSS P25774 1/20 0.37
LMNA P02545 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HTT P42858 2/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6415706 0.88 FAAH (0.42) FAAHHDAC3HDAC4HDAC1HDAC7
SCHEMBL6206684 0.83 NPC1 (0.42) FAAHRAB9ANPC1CTSSLMNA
SCHEMBL6206918 0.81 METAP2 (0.40) FAAHRAB9ANPC1CTSSLMNA
Hydrochloric Acid SCHEMBL5946008 0.80 CTSS (0.42) RAB9ANPC1CTSS
SCHEMBL14974258 0.79 PTPN2 (0.41) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5516626 0.78 HDAC3 (0.40) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6415401 0.76 REN (0.42) CTSSLMNASMN1; SMN2HTTTSHR
SCHEMBL5516628 0.75 TSHR (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5475660 0.74 TSHR (0.35) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5475666 0.74 TSHR (0.35) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1503997-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-02-09 EP disclosed
WO-2003097617-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2003-11-27 WO disclosed