SCHEMBL6207396

SCHEMBL6207396

CC(Oc1cnccn1)c1cc(NC(=O)Nc2nc(C(C)(C)C)cs2)ccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
POLB P06746 1/20 0.47
BRAF P15056 2/20 0.44
FLT3 P36888 1/20 0.42
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
RET P07949 1/20 0.40
GAA P10253 1/20 0.39
FFAR2 O15552 1/20 0.38
ROCK1 Q13464 1/20 0.37
SMARCA2 P51531 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080568 0.83 KMT2A (0.48) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL6207387 0.81 KMT2A (0.47) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL6240758 0.78 RAB9A (0.49) MEN1KMT2ANPC1RAB9AMAPK1
SCHEMBL6257230 0.72 MEN1 (0.43) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL22103784 0.69 RAB9A (0.76) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL22125497 0.68 SMARCA2 (0.72) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL14014120 0.68 RAB9A (0.80) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL20788543 0.68 NPC1 (0.77) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL6079119 0.67 ALDH1A1 (0.52) MEN1KMT2AALDH1A1MAPK1SMN1; SMN2
SCHEMBL10078887 0.66 MEN1 (1.00) MEN1KMT2ANPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1545523-A1 3-&-grave;(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES ASP38 MAP KINASE INHIBITORS Astex Technology Limited (GB) 2005-06-29 EP disclosed
WO-2004004720-A1 3-`(HETERO) ARYLMETHOXY ! PYRIDINES AND THEIR ANALOGUES AS P38 MAP KINASE INHIBITORS ASTEX TECHNOLOGY LIMITED (GB) 2004-01-15 WO disclosed