SCHEMBL6208577

SCHEMBL6208577

Cc1cc(CC(=O)OC(C)(C)C)ccc1N(C(N)=O)c1ccccc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
EPHX2 P34913 1/20 0.32
PDK2 Q15119 1/20 0.32
PPARG P37231 3/20 0.32
PPARA Q07869 2/20 0.32
RIPK1 Q13546 1/20 0.31
RIPK3 Q9Y572 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
TP53 P04637 1/20 0.31
POLQ O75417 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6037550 0.80 MTNR1A (0.50) MTNR1AMTNR1BLMNAPOLBALDH1A1
SCHEMBL5152274 0.74 GAA (0.45) LMNAALDH1A1
SCHEMBL5331837 0.74 LMNA (0.42) LMNAPOLBALDH1A1POLQ
SCHEMBL5155096 0.72 POLB (0.55) LMNAPOLBITGB1ITGA4ALDH1A1
SCHEMBL5281926 0.71 MTNR1A (0.49) MTNR1AMTNR1BLMNAPOLBALDH1A1
SCHEMBL6964628 0.69 GAA (0.46) LMNAPOLBALDH1A1
SCHEMBL2432439 0.69 ALDH1A1 (0.45) MTNR1AMTNR1BPPARGRIPK1RIPK3
SCHEMBL27478926 0.68 TRPM8 (0.38) LMNAALDH1A1TP53
SCHEMBL20566969 0.68 IDO1 (0.50) MTNR1AMTNR1BLMNAPPARGPPARA
SCHEMBL17102979 0.67 LMNA (0.37) LMNAALDH1A1POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189612-A4 VLA-4 INHIBITOR COMPOUNDS DAIICHI SEIYAKU CO (JP) 2005-02-16 EP disclosed
EP-1189612-A1 VLA-4 INHIBITOR COMPOUNDS Daiichi Pharmaceutical Co., Ltd. (JP) 2002-03-27 EP disclosed
WO-2001000206-A1 VLA-4 INHIBITOR COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-04 WO disclosed