SCHEMBL6208701

SCHEMBL6208701

CC(C)CC(OCc1cc(N2CCN(C(=O)O)CC2)ccc1-c1ccccc1)C(=O)NCC#N

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 15/20 0.48
CTSK P43235 15/20 0.48
CTSB P07858 14/20 0.48
CTSL P07711 14/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210052 0.83 CTSK (0.57) CTSSCTSKCTSBCTSL
SCHEMBL4699481 0.83 CTSS (0.51) CTSSCTSKCTSBCTSL
SCHEMBL4700794 0.82 CTSS (0.62) CTSSCTSKCTSBCTSL
SCHEMBL4700947 0.81 CTSL (0.66) CTSSCTSKCTSBCTSL
SCHEMBL6208704 0.80 CTSK (0.41) CTSSCTSKCTSBCTSL
SCHEMBL4700791 0.79 CTSS (0.45) CTSSCTSKCTSBCTSL
SCHEMBL6208357 0.79 CTSK (0.60) CTSSCTSKCTSBCTSL
SCHEMBL6209030 0.77 CTSS (0.53) CTSSCTSKCTSBCTSL
SCHEMBL6001121 0.75 CTSB (0.53) CTSSCTSKCTSBCTSL
SCHEMBL4699860 0.74 CTSK (0.72) CTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-A4 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-10-12 EP disclosed
EP-1372655-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada & Co. (CA) 2004-01-02 EP disclosed
WO-2002069901-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2002-09-12 WO disclosed