SCHEMBL6208713

SCHEMBL6208713

NC(=O)CCCC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.36
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
F10 P00742 3/20 0.34
F2 P00734 1/20 0.34
PRSS1 P07477 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
TPSAB1 Q15661 1/20 0.33
TPSD1 Q9BZJ3 1/20 0.33
TPSG1 Q9NRR2 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TSHR P16473 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
DPP4 P27487 1/20 0.32
LMNA P02545 1/20 0.32
ESR1 P03372 1/20 0.32
STS P08842 1/20 0.32
RECQL P46063 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046219 0.86 PARP1 (0.35) PARP1F10F2PRSS1L3MBTL1
SCHEMBL6209846 0.86 DPP4 (0.35) PARP1KDM4EHTTF10F2
SCHEMBL6209170 0.86 PARP1 (0.35) PARP1KDM4EHTTF10F2
SCHEMBL6209393 0.86 CTSL (0.36)
SCHEMBL6209760 0.83 MT-CO2 (0.33) L3MBTL1MEN1KMT2ADPP4
SCHEMBL6210370 0.83 FKBP1A (0.41) PARP1ALDH1A1TSHR
SCHEMBL6210338 0.81 DPP4 (0.46) TSHRGAADPP4
SCHEMBL4045821 0.80 PARP1 (0.35) PARP1F10F2PRSS1ALDH1A1
SCHEMBL4042325 0.80 DPP4 (0.40) PARP1KDM4EF10F2PRSS1
SCHEMBL4045826 0.80 TSHR (0.35) PARP1KDM4EF10F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed