SCHEMBL6210370

SCHEMBL6210370

NC(=O)CCCC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 1/20 0.41
SMYD3 Q9H7B4 2/20 0.39
ALDH1A1 P00352 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
VNN1 O95497 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043418 0.87 FKBP1A (0.38) FKBP1ASMYD3ALDH1A1CYP2C9TSHR
SCHEMBL6210568 0.86 SMYD3 (0.38) FKBP1ASMYD3ALDH1A1CYP2C9TSHR
SCHEMBL6209144 0.86 SMYD3 (0.38) FKBP1ASMYD3ALDH1A1CYP2C9TSHR
SCHEMBL6208880 0.86 KDM4E (0.42) FKBP1ASMYD3ALDH1A1TSHRCYP2C19
SCHEMBL6208973 0.84 TBXAS1 (0.35) ALDH1A1VNN1
SCHEMBL6210597 0.83 PARP1 (0.40) ALDH1A1CYP2C9PARP1PARP2VNN1
SCHEMBL6208713 0.83 PARP1 (0.36) ALDH1A1TSHRPARP1
SCHEMBL6210118 0.82 DPP4 (0.44) SMYD3ALDH1A1CYP2C9CYP2C19
SCHEMBL6211755 0.81 DPP4 (0.45) SMYD3ALDH1A1
SCHEMBL4046437 0.81 FKBP1A (0.41) FKBP1ASMYD3VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed