SCHEMBL6208960

SCHEMBL6208960

Cc1nsc(N[C@@H](CC(C)C)C(=O)NCC#N)c1-c1ccccc1C1CNCCN1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 15/20 0.48
CTSS P25774 14/20 0.48
CTSB P07858 13/20 0.48
CTSK P43235 10/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701917 0.87 CTSL (0.47) CTSLCTSSCTSBCTSK
SCHEMBL4699307 0.78 CTSL (0.60) CTSLCTSSCTSBCTSK
SCHEMBL4701389 0.78 CTSL (0.52) CTSLCTSSCTSBCTSK
SCHEMBL4702155 0.76 CTSL (0.69) CTSLCTSSCTSBCTSK
SCHEMBL4702170 0.76 CTSL (0.69) CTSLCTSSCTSBCTSK
SCHEMBL4698847 0.76 CTSB (0.55) CTSLCTSSCTSBCTSK
SCHEMBL4699683 0.74 CTSL (0.51) CTSLCTSSCTSBCTSK
SCHEMBL6909712 0.74 CTSS (0.39) CTSLCTSSCTSBCTSK
SCHEMBL4701283 0.73 CTSL (0.54) CTSLCTSSCTSBCTSK
SCHEMBL4704047 0.73 CTSL (0.54) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-A4 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-10-12 EP disclosed
EP-1372655-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada & Co. (CA) 2004-01-02 EP disclosed
WO-2002069901-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2002-09-12 WO disclosed