SCHEMBL6209099

SCHEMBL6209099

O=C(NCCCCC(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)c1ccc(-c2cnco2)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.41
PTAFR P25105 9/20 0.41
ALDH1A1 P00352 1/20 0.40
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
TAOK1 Q7L7X3 1/20 0.36
DPP4 P27487 1/20 0.36
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6215209 0.88 ROCK2 (0.40) ROCK2PTAFRALDH1A1DPP4
SCHEMBL6212956 0.88 ROCK2 (0.41) ROCK2PTAFROPRM1OPRD1OPRK1
SCHEMBL6209605 0.87 DPP4 (0.44) PTAFRALDH1A1DPP4NAMPT
SCHEMBL5941500 0.86 NAMPT (0.46) PTAFRALDH1A1DPP4NAMPT
SCHEMBL6209860 0.86 HDAC1 (0.44) PTAFRDPP4
SCHEMBL6211981 0.85 ALDH1A1 (0.46) PTAFRALDH1A1NAMPT
SCHEMBL6212212 0.85 PTAFR (0.42) PTAFRALDH1A1
SCHEMBL6211236 0.85 PTAFR (0.40) PTAFRALDH1A1NAMPT
SCHEMBL6212722 0.85 CHRM4 (0.43) PTAFRDPP4NAMPT
SCHEMBL6212663 0.84 TAOK1 (0.39) ROCK2ALDH1A1TAOK1DPP4NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed