SCHEMBL6209860

SCHEMBL6209860

O=C(NCCCCC(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)c1ccc(-c2cccs2)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.44
HDAC3 O15379 2/20 0.44
CHRM4 P08173 1/20 0.43
PTAFR P25105 7/20 0.41
DPP4 P27487 1/20 0.40
PREP P48147 1/20 0.40
DRD2 P14416 4/20 0.39
DRD4 P21917 3/20 0.39
HTR2A P28223 1/20 0.39
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
RAD52 P43351 1/20 0.37
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210236 0.88 CHRM4 (0.41) HDAC1HDAC3CHRM4PTAFRDPP4
SCHEMBL6210587 0.88 HDAC1 (0.42) HDAC1HDAC3CHRM4PTAFRDPP4
SCHEMBL5941500 0.88 NAMPT (0.46) CHRM4PTAFRDPP4
SCHEMBL6209605 0.87 DPP4 (0.44) HDAC1HDAC3PTAFRDPP4
SCHEMBL6209099 0.86 ROCK2 (0.41) PTAFRDPP4
SCHEMBL6212212 0.85 PTAFR (0.42) PTAFR
SCHEMBL6211236 0.85 PTAFR (0.40) HDAC1HDAC3CHRM4PTAFRDRD2
SCHEMBL6212722 0.85 CHRM4 (0.43) CHRM4PTAFRDPP4
SCHEMBL6211981 0.84 ALDH1A1 (0.46) HDAC1HDAC3PTAFRDRD2HTR2A
SCHEMBL6259166 0.83 NAMPT (0.41) HDAC1HDAC3CHRM4PTAFRPREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed