SCHEMBL6209944

SCHEMBL6209944

CCc1nc(CC)nc(-c2cc(C)c(C)cc2O)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
G6PD P11413 1/20 0.39
CYP2C9 P11712 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
CCR6 P51684 1/20 0.39
HIF1A Q16665 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 4/20 0.37
TDP1 Q9NUW8 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6512115 0.76 ALDH1A1 (0.46) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL9637931 0.72 MAPK1 (0.58) MAPTALDH1A1KDM4EHPGDALOX15
SCHEMBL9486648 0.71 ALDH1A1 (0.43) MAPTALDH1A1KDM4EPKMHPGD
SCHEMBL6243491 0.70 ALDH1A1 (0.72) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL15890818 0.67
SCHEMBL15131515 0.64 ADORA3 (0.41) ALDH1A1CYP1A2MAPK1CYP2C19NPSR1
SCHEMBL616464 0.64 TSPO (0.34) ALDH1A1KDM4EMAPK1LMNATSHR
SCHEMBL2614743 0.64 HRH4 (0.33)
Formaldehyde SCHEMBL7997140 0.64 ALDH1A1 (0.62) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL26437128 0.64 ALDH1A1 (0.79) MAPTALDH1A1KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115937-B1 AQUEOUS COMPOSITIONS OF UV-ACTIVE AGENTS, THEIR PRODUCTION AND USE CLARIANT FINANCE BVI LTD (VG) 2005-03-02 EP disclosed
EP-0834304-B1 Use of liposomogenic UV absorbers to protect hair CIBA SC HOLDING AG (CH) 2005-01-26 EP disclosed
US-6780827-B1 TEXTILE FINISHING; INCLUDING CARBOXYL CONTAINING CROSSLINKED COPOLYMER TO PREVENT PRESSURE BUILDUP OR DYE OR BRIGHTENER FILTRATION DEPOSITS CLARIANT FINANCE (BVI) LIMITED (VG) 2004-08-24 US disclosed
US-6723256-B1 DISPERSANT SYSTEM CONTAINING SUCH AS PHENOLIC NOVOLAK-METHYLATED POLYETHYLENE GLYCOL COPOLYMER, ALKYLSULPHONATE, AND MALEIC ANHYDRIDE-METHYL VINYL ETHER-1,9-DECADIENE TERPOLYMER; STABILITY CLARIANT FINANCE (BVI) LIMITED (VG) 2004-04-20 US disclosed
EP-1115938-B1 AQUEOUS COMPOSITIONS OF UV-ACTIVE AGENTS, THEIR PRODUCTION AND USE CLARIANT FINANCE BVI LTD (VG) 2003-06-04 EP disclosed
EP-1115938-A1 AQUEOUS COMPOSITIONS OF UV-ACTIVE AGENTS, THEIR PRODUCTION AND USE Clariant Finance (BVI) Limited (VG) 2001-07-18 EP disclosed
EP-0815071-B1 LIPOSOMOGENIC UV ABSORBERS CIBA SC HOLDING AG (CH) 2001-04-11 EP disclosed
WO-2000011257-A1 AQUEOUS COMPOSITIONS OF UV-ACTIVE AGENTS, THEIR PRODUCTION AND USE CLARIANT FINANCE (BVI) LIMITED (VG) 2000-03-02 WO disclosed
US-6017556-A PROTECTING HUMAN HAIR FROM THE DAMAGING EFFECT OF ULTRAVIOLET RADIATION BY TREATING HUMAN HAIR WITH A LIPOSOMOGENIC ULTRAVIOLET RADIATION ABSORBER CIBA SPECIALTY CHEMICALS CORPORATION (US) 2000-01-25 US disclosed
US-6015575-A TRIAZINE, BENZOTRIAZOLE, BENZOPHENONE AND AMINOBENZOIC ACID DERIVATIVES AS RADIATION ABSORBERS CIBA SPECIALTY CHEMICALS CORPORATION (US) 2000-01-18 US disclosed
EP-0468921-B2 Aqueous dispersions of slightly soluble UV absorbing agents CIBA GEIGY AG (CH) 1998-07-22 EP disclosed
EP-0834304-A2 Liposomogenic UV absorbers Ciba SC Holding AG (CH) 1998-04-08 EP disclosed
US-5575958-A HYDROXYPHENYL TRIAZINES CIBA-GEIGY CORPORATION (US) 1996-11-19 US disclosed
EP-0523006-B1 Process for printing and photochemically stabilizing polyester fibre materials CIBA GEIGY AG (CH) 1995-11-29 EP disclosed
EP-0523006-A1 Process for printing and photochemically stabilizing polyester fibre materials CIBA-GEIGY AG (CH) 1993-01-13 EP disclosed
EP-0280653-B1 PROCESS FOR IMPROVING THE PHOTOCHEMICAL STABILITY OF DYEINGS ON FIBROUS POLYESTER MATERIALS CIBA-GEIGY AG (CH) 1992-05-13 EP disclosed
EP-0468921-A1 Aqueous dispersions of slightly soluble UV absorbing agents CIBA-GEIGY AG (CH) 1992-01-29 EP disclosed
US-4831068-A PHENYL-S-TRIAZINE DERIVATIVES AS UV ABSORBERS CIBA-GEIGY CORPORATION (US) 1989-05-16 US disclosed