SCHEMBL6209952

SCHEMBL6209952

CC(C)C[C@@H](Oc1cccc(-c2ccc(N3CCNCC3)cc2)c1)C(=O)NCC#N

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.71
CTSL P07711 16/20 0.71
CTSB P07858 15/20 0.71
CTSK P43235 15/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698932 1.00 CTSS (0.71) CTSSCTSLCTSBCTSK
SCHEMBL4701781 0.92 CTSL (0.68) CTSSCTSLCTSBCTSK
SCHEMBL6208357 0.89 CTSK (0.60) CTSSCTSLCTSBCTSK
SCHEMBL4700960 0.87 CTSS (0.68) CTSSCTSLCTSBCTSK
SCHEMBL6208955 0.87 CTSS (0.68) CTSSCTSLCTSBCTSK
SCHEMBL6208924 0.85 CTSK (0.59) CTSSCTSLCTSBCTSK
SCHEMBL4699757 0.85 CTSK (0.59) CTSSCTSLCTSBCTSK
SCHEMBL4698729 0.84 CTSK (0.64) CTSSCTSLCTSBCTSK
SCHEMBL4699494 0.84 CTSL (0.71) CTSSCTSLCTSBCTSK
SCHEMBL4699463 0.84 CTSL (0.68) CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-A4 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-10-12 EP disclosed
EP-1372655-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada & Co. (CA) 2004-01-02 EP disclosed
WO-2002069901-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2002-09-12 WO disclosed