SCHEMBL6210568

SCHEMBL6210568

CC(C)(CC(N)=O)CC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.38
FKBP1A P62942 1/20 0.38
ALDH1A1 P00352 2/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
PARP1 P09874 1/20 0.34
PARP2 Q9UGN5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208666 0.87 KDM4E (0.39) SMYD3ALDH1A1TSHRCYP2C19
SCHEMBL6210370 0.86 FKBP1A (0.41) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL6209144 0.85 SMYD3 (0.38) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL6210592 0.84 PAX8 (0.40) FKBP1AALDH1A1CYP2C9PARP1PARP2
SCHEMBL6209170 0.84 PARP1 (0.35) FKBP1AALDH1A1TSHRPARP1
SCHEMBL4044948 0.82 SMYD3 (0.38) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL4044950 0.81 DPP4 (0.39) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL4043418 0.80 FKBP1A (0.38) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL4038231 0.79 SMYD3 (0.39) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL6210371 0.79 CTSK (0.38) SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed