SCHEMBL6211580

SCHEMBL6211580

O=C(NCCCCC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.43
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
PPARD Q03181 2/20 0.39
CHRM4 P08173 1/20 0.39
CXCR3 P49682 2/20 0.39
PTAFR P25105 1/20 0.38
TRPV1 Q8NER1 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
SMYD3 Q9H7B4 2/20 0.37
SLC6A5 Q9Y345 1/20 0.37
GCGR P47871 2/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211755 0.92 DPP4 (0.45) NAMPTPPARDPTAFRSMYD3SLC6A5
SCHEMBL6210722 0.90 CHRM4 (0.42) NAMPTCHRM4PTAFRDPP4
SCHEMBL6258369 0.90 LMNA (0.44) NAMPTCHRM2CHRM1PPARDCHRM4
SCHEMBL6210118 0.89 DPP4 (0.44) NAMPTPTAFRHDAC3HDAC1SMYD3
SCHEMBL6275935 0.88 NAMPT (0.41) NAMPTCHRM2CHRM1PPARDCHRM4
SCHEMBL6259166 0.87 NAMPT (0.41) NAMPTCHRM2CHRM1CHRM4CXCR3
SCHEMBL6211528 0.85 ALDH1A1 (0.44) NAMPTPTAFRHDAC3HDAC1SMYD3
SCHEMBL6210861 0.85 HDAC1 (0.41) NAMPTPTAFRHDAC3HDAC1SMYD3
SCHEMBL6210587 0.84 HDAC1 (0.42) CHRM4PTAFRHDAC3HDAC1DPP4
SCHEMBL6215209 0.84 ROCK2 (0.40) PTAFRSMYD3DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed