SCHEMBL6210587

SCHEMBL6210587

O=C(NCCCCC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)c1ccc(-c2cccs2)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.42
HDAC3 O15379 2/20 0.42
CHRM4 P08173 1/20 0.41
PTAFR P25105 7/20 0.39
DPP4 P27487 2/20 0.38
PREP P48147 1/20 0.38
DRD2 P14416 3/20 0.37
DRD4 P21917 3/20 0.37
HTR2A P28223 1/20 0.37
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210489 0.88 CHRM4 (0.39) HDAC1HDAC3CHRM4DPP4PREP
SCHEMBL6211755 0.88 DPP4 (0.45) PTAFRDPP4
SCHEMBL6210118 0.88 DPP4 (0.44) HDAC1HDAC3PTAFRDPP4
SCHEMBL6209860 0.88 HDAC1 (0.44) HDAC1HDAC3CHRM4PTAFRDPP4
SCHEMBL6215209 0.86 ROCK2 (0.40) PTAFRDPP4
SCHEMBL6210861 0.86 HDAC1 (0.41) HDAC1HDAC3PTAFRHTR2AHDAC2
SCHEMBL6210722 0.85 CHRM4 (0.42) CHRM4PTAFRDPP4
SCHEMBL6211528 0.85 ALDH1A1 (0.44) HDAC1HDAC3PTAFRHTR2A
SCHEMBL6211580 0.84 NAMPT (0.43) HDAC1HDAC3CHRM4PTAFRDPP4
SCHEMBL4042901 0.82 CTSK (0.47) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed