SCHEMBL6213602

SCHEMBL6213602

C[C@@H]1CC[C@H](N(C(=O)C2(NC(=O)c3cc4ccccc4o3)CCCCC2)S(=O)(=O)c2ccccn2)[C@@H](O)CN1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 17/20 0.39
CTSL P07711 13/20 0.37
CTSS P25774 10/20 0.37
CTSB P07858 5/20 0.37
CTSV O60911 2/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604880 0.88 CTSK (0.39) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6211960 0.88 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6211256 0.84 RAB9A (0.31) NPC1TP53RAB9ASMN1; SMN2
SCHEMBL6603823 0.80 PSEN1 (0.30)
SCHEMBL6673927 0.80 CTSK (0.39) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6601357 0.80 HDAC3 (0.31) POLB
SCHEMBL6601633 0.79 PTGDR2 (0.31)
SCHEMBL6212431 0.73 RAB9A (0.31) CTSKCTSLCTSSNPC1TP53
SCHEMBL6843807 0.72 CTSK (0.51) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6214202 0.72 CTSK (0.47) CTSKCTSLCTSSCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307203-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2005-08-17 EP claimed
EP-1392657-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-03-10 EP claimed
EP-1392657-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2004-03-03 EP claimed
WO-2003053331-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-07-03 WO claimed
EP-1307203-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-05-07 EP claimed
WO-2001070232-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-09-27 WO claimed
EP-1307203-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2005-08-17 EP disclosed
EP-1392657-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-03-10 EP disclosed
EP-1392657-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2004-03-03 EP disclosed
WO-2003053331-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-07-03 WO disclosed
EP-1307203-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-05-07 EP disclosed
WO-2001070232-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-09-27 WO disclosed