SCHEMBL6218809

SCHEMBL6218809

CC(C)(CO)c1ccn2ccnc2n1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
GABRA1 P14867 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31
GABRA3 P34903 2/20 0.31
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCNA1 P78396 1/20 0.30
CDK5 Q00535 1/20 0.30
DYRK1A Q13627 1/20 0.30
CDK5R1 Q15078 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5769993 0.81 GABRA1 (0.39) NPC1RAB9AGABRA1GABRG2GABRB3
SCHEMBL5770463 0.81 ALDH1A1 (0.36) NPC1RAB9ADYRK1A
SCHEMBL5768555 0.78 GABRA1 (0.33) NPC1RAB9AGABRA1GABRG2GABRB3
SCHEMBL5771081 0.77 KDM4E (0.34) NPC1RAB9AGABRA1GABRG2GABRB3
SCHEMBL5770695 0.74 JAK2 (0.36)
SCHEMBL6217363 0.73 PLCG1 (0.38) NPC1RAB9A
SCHEMBL5771074 0.70 CCR1 (0.38) NPC1RAB9ADYRK1A
SCHEMBL22726577 0.68 SSTR4 (0.46) CDK2
SCHEMBL6102107 0.67 ALDH1A1 (0.39) NPC1RAB9ADYRK1A
SCHEMBL5808966 0.67 RAB9A (0.39) NPC1RAB9ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381606-B1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2005-07-20 EP disclosed