SCHEMBL622416

SCHEMBL622416

CC(C)[C@H](NC(=O)CCc1ccc(O)cc1)C(=O)NC(C=O)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSB P07858 4/20 0.54
GRIA1 P42261 1/20 0.50
CTSD P07339 1/20 0.46
ACE P12821 1/20 0.45
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
CASP1 P29466 2/20 0.44
TRPV1 Q8NER1 1/20 0.44
IL1B P01584 1/20 0.43
CASP3 P42574 1/20 0.43
CASP7 P55210 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623362 0.94 CTSB (0.58) CTSBCTSDACECASP1IL1B
SCHEMBL621818 0.91 CTSB (0.53) CTSBCTSDACECASP1IL1B
SCHEMBL623363 0.90 CTSB (0.53) CTSBCTSDCASP1IL1B
SCHEMBL10084539 0.90 CTSB (0.53) CTSBCTSDCASP1
SCHEMBL621711 0.89 CTSB (0.54) CTSBACE
SCHEMBL623793 0.89 ALDH1A1 (0.54) CTSBCTSDCASP1
SCHEMBL10084534 0.89 CTSB (0.51) CTSBCTSDCASP1IL1B
SCHEMBL623259 0.88 CTSB (0.53) CTSBCTSDCASP1
SCHEMBL622188 0.86 CTSB (0.48) CTSBCTSDCASP1IL1B
SCHEMBL10084540 0.85 CTSB (0.48) CTSBCTSDTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed