SCHEMBL623259

SCHEMBL623259

CC(C)[C@H](NC(=O)CCc1ccc(C(F)(F)F)cc1)C(=O)NC(C=O)Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.53
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50
FFAR2 O15552 1/20 0.49
CTSL P07711 1/20 0.46
CASP1 P29466 1/20 0.44
CTSD P07339 1/20 0.44
PLAAT3 P53816 1/20 0.43
PLAAT5 Q96KN8 1/20 0.43
PLAAT2 Q9NWW9 1/20 0.43
PLAAT4 Q9UL19 1/20 0.43
UTS2R Q9UKP6 2/20 0.42
HTRA1 Q92743 1/20 0.42
PDPK1 O15530 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623362 0.91 CTSB (0.58) CTSBCASP1CTSD
SCHEMBL10084323 0.90 CTSB (0.48) CTSBCYP1A2CYP3A4CYP2C9TSHR
SCHEMBL623363 0.89 CTSB (0.53) CTSBCTSLCASP1CTSD
SCHEMBL622416 0.88 CTSB (0.54) CTSBCASP1CTSD
SCHEMBL621818 0.88 CTSB (0.53) CTSBCASP1CTSDUTS2R
SCHEMBL10084539 0.87 CTSB (0.53) CTSBCASP1CTSDUTS2RHTRA1
SCHEMBL10084535 0.85 CTSB (0.47) CTSBCASP1CTSDHTRA1
SCHEMBL621459 0.85 CTSB (0.46) CTSBCASP1CTSDHTRA1
SCHEMBL623793 0.85 ALDH1A1 (0.54) CTSBCASP1CTSD
SCHEMBL10084534 0.85 CTSB (0.51) CTSBCASP1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed
WO-2012021788-A2 DIPEPTIDE CALPAIN INHIBITORS BANYAN BIOMARKERS (US) 2012-02-16 WO disclosed