SCHEMBL6228337

SCHEMBL6228337

CCCNC(=O)Nc1nc2ccccc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 11/20 1.00
RAB9A P51151 11/20 1.00
SMN1; SMN2 Q16637 9/20 0.85
ADORA1 P30542 1/20 0.62
DYRK1A Q13627 1/20 0.62
NFKB1 P19838 3/20 0.62
NFKB2 Q00653 3/20 0.62
RELA Q04206 3/20 0.62
MAPT P10636 3/20 0.62
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
GAA P10253 2/20 0.62
ALDH1A1 P00352 3/20 0.60
STAT1 P42224 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2C19 P33261 1/20 0.60
MAPK1 P28482 2/20 0.59
KDM4E B2RXH2 2/20 0.59
HTT P42858 1/20 0.59
ACP1 P24666 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6229810 0.92 NPC1 (1.00) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL31041 0.91 NPC1 (0.93) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL1842324 0.89 NPC1 (1.00) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL2792307 0.87 NPC1 (0.78) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
Hydrochloric Acid SCHEMBL1844043 0.87 NPC1 (0.97) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL2792818 0.85 NPC1 (0.74) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL2791120 0.85 RAB9A (0.74) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL2816736 0.84 RAB9A (0.72) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL6905516 0.84 RAB9A (0.72) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A
SCHEMBL27634788 0.83 NPC1 (0.84) NPC1RAB9ASMN1; SMN2ADORA1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3102203-A2 ANTIBACTERIAL COMBINATIONS COMPRISING POLYMYXIN SPERO GYRASE, INC. (US) 2016-12-14 EP disclosed
WO-2015114452-A2 ANTIBACTERIAL COMPOUNDS BIOTA EUROPE LTD (GB) 2015-08-06 WO disclosed
US-6900219-B2 ABCA-1 elevating compounds CV THERAPEUTICS, INC. (US) 2005-05-31 US disclosed
EP-1513534-A2 COMPOUNDS FOR INCREASING ABCA-1 EXPRESSION USEFUL FOR TREATING CORONARY ARTERY DISEASE AND ATHEROSCLEROSIS CV THERAPEUTICS, INC. (US) 2005-03-16 EP disclosed
US-20030220356-A1 ABCA-1 elevating compounds CV THERAPEUTICS, INC. 2003-11-27 US disclosed
WO-2003084544-A2 COMPOUNDS DOR INCREASING ABCA-1 EXPRESSION USEFUL FOR TREATING CORONARY ARTERY DISEASE AND ATHEROSCLEROSIS CV THERAPEUTICS, INC. (US) 2003-10-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030220356-A1 ABCA-1 elevating compounds ABCD3, ABCE1, ABCB4 NPC1 6/4885RAB9A 2138/4885SMN1; SMN2 4558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.