SCHEMBL6231990

SCHEMBL6231990

Nc1ccc2sc(C(=O)N3CCC(c4ccccc4)CC3)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CHRNA7 P36544 1/20 0.47
SCD5 Q86SK9 3/20 0.46
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PRSS12 P56730 1/20 0.46
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 1/20 0.46
CCR1 P32246 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CAPN1 P07384 1/20 0.44
CTSB P07858 1/20 0.44
SPR P35270 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6252866 0.83 ALDH1A1 (0.68) HRH4L3MBTL1SCD5NPC1MAPT
SCHEMBL6253982 0.81 ALDH1A1 (0.57) HRH4L3MBTL1MAPTCA12CA1
SCHEMBL6232921 0.80 ALDH1A1 (0.66) HRH4L3MBTL1CHRNA7CA12CA1
SCHEMBL6234648 0.80 CHRNA7 (0.53) HRH4L3MBTL1CHRNA7NPC1RAB9A
SCHEMBL6254206 0.80 CHRNA7 (0.53) HRH4L3MBTL1CHRNA7NPC1RAB9A
SCHEMBL6616703 0.79 ALDH1A1 (0.51) HRH4L3MBTL1CHRNA7RAB9ACA12
SCHEMBL6234089 0.78 HRH4 (0.69) HRH4L3MBTL1CHRNA7NPC1RAB9A
SCHEMBL6231088 0.78 L3MBTL1 (0.69) HRH4L3MBTL1CHRNA7NPC1MAPT
SCHEMBL4395877 0.76 TPSAB1 (0.55) HRH4L3MBTL1CA12CA1CA2
SCHEMBL13212972 0.74 CA12 (0.71) NPC1RAB9ASMN1; SMN2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed