SCHEMBL623207

SCHEMBL623207

FC(F)(F)Oc1cccc(-c2cn3nc(N4CCC5(CCNCC5)C4)sc3n2)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 6/20 0.48
F2RL3 Q96RI0 4/20 0.40
PIM3 Q86V86 2/20 0.39
FLT3 P36888 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
THRB P10828 2/20 0.38
SCN4A P35499 1/20 0.38
SCN9A Q15858 1/20 0.38
MAPT P10636 2/20 0.38
TYRO3 Q06418 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
XDH P47989 1/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
MGLL Q99685 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623949 0.95 PIM1 (0.47) PIM1F2RL3PIM3FLT3PIM2
SCHEMBL624740 0.91 PIM1 (0.48) PIM1F2RL3PIM3PIM2THRB
SCHEMBL623996 0.85 THRB (0.42) PIM1F2RL3THRBMAPTHCRTR1
SCHEMBL623206 0.84 PIM1 (0.47) PIM1
SCHEMBL625255 0.83 PIM3 (0.48) PIM1F2RL3PIM3PIM2THRB
SCHEMBL625249 0.81 PIM2 (0.48) PIM1F2RL3PIM3PIM2THRB
SCHEMBL624528 0.81 CYP3A4 (0.41) THRBMAPTHCRTR1HCRTR2RXFP1
SCHEMBL625561 0.80 PIM1 (0.49) PIM1F2RL3PIM3FLT3PIM2
SCHEMBL625512 0.79 THRB (0.44) PIM1F2RL3THRBMAPTRXFP1
SCHEMBL623867 0.79 PIM1 (0.44) PIM1F2RL3THRBMAPTXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed