SCHEMBL6232865

SCHEMBL6232865

CCCC(NC(=O)c1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 8/20 0.46
TAS1R1 Q7RTX1 8/20 0.46
TSHR P16473 1/20 0.39
CTSK P43235 2/20 0.39
MCHR1 Q99705 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
LMNA P02545 4/20 0.36
MAPT P10636 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PTBP1 P26599 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235078 0.92 CTSK (0.48) TAS1R3TAS1R1TSHRCTSKCYP1A2
SCHEMBL4048294 0.88 ALDH1A1 (0.37) TAS1R3TAS1R1TSHRMCHR1CYP1A2
SCHEMBL6274440 0.88 CTSK (0.48) CTSKALDH1A1KMT2A
SCHEMBL4045150 0.88 CTSK (0.44) CTSKLMNAALDH1A1KMT2A
SCHEMBL4038812 0.86 CTSK (0.54) CTSK
SCHEMBL4039713 0.86 CTSK (0.45) CTSK
SCHEMBL4042617 0.85 CTSK (0.46) TAS1R3TAS1R1CTSK
SCHEMBL4040752 0.85 CTSK (0.54) CTSKALDH1A1
SCHEMBL4044103 0.85 CTSK (0.42) TAS1R3TAS1R1CTSKKMT2A
SCHEMBL4042168 0.85 CTSK (0.42) CTSKLMNASMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed