SCHEMBL4048294

SCHEMBL4048294

CCCC(NC(=O)Oc1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
TSHR P16473 3/20 0.37
HPGD P15428 1/20 0.37
KCNQ1 P51787 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
CHRM5 P08912 1/20 0.34
MAPT P10636 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
BMP1 P13497 1/20 0.32
KMT2A Q03164 1/20 0.32
MCHR1 Q99705 1/20 0.32
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047459 0.93 CTSK (0.38) ALDH1A1TSHRHPGDKCNQ1TAS1R3
SCHEMBL4050306 0.89 PKM (0.36) ALDH1A1TSHRHPGDKCNQ1TAS1R3
SCHEMBL4045249 0.89 CTSK (0.36) HPGDLMNA
SCHEMBL4050093 0.89 HTT (0.41) ALDH1A1TSHRHPGDKCNQ1TAS1R3
SCHEMBL6232865 0.88 TAS1R3 (0.46) ALDH1A1TSHRTAS1R3TAS1R1MAPT
SCHEMBL4044695 0.88 CTSK (0.36)
SCHEMBL4048544 0.86 P2RY12 (0.32)
SCHEMBL4051941 0.85 ELOVL6 (0.38) TSHRLMNASMN1; SMN2
SCHEMBL4043292 0.85 ALDH1A1 (0.37) ALDH1A1CHRM5MAPTLMNA
SCHEMBL4047785 0.85 CTSK (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed