SCHEMBL6233612

SCHEMBL6233612

CN(C)c1nc2cc([N+](=O)[O-])ccc2n1CCCO

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 4/20 0.48
MAP4K4 O95819 2/20 0.46
CSNK1D P48730 2/20 0.46
CLK2 P49760 2/20 0.46
IRAK1 P51617 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
DYRK3 O43781 1/20 0.46
ROCK2 O75116 1/20 0.46
RPS6KA5 O75582 1/20 0.46
PRKD3 O94806 1/20 0.46
CDK1 P06493 1/20 0.46
PHKG2 P15735 1/20 0.46
MARK3 P27448 1/20 0.46
CSNK1A1 P48729 1/20 0.46
GSK3B P49841 1/20 0.46
NEK4 P51957 1/20 0.46
CSNK1G2 P78368 1/20 0.46
ITK Q08881 1/20 0.46
MAP4K2 Q12851 1/20 0.46
DYRK1A Q13627 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230911 0.93 MAPT (0.50) IRAK4PKMALDH1A1MAPTPOLB
SCHEMBL6231609 0.84 KMT2A (0.51) IRAK4MAP4K4CSNK1DCLK2IRAK1
SCHEMBL6277473 0.83 MAPT (0.47) IRAK4MAP4K4CSNK1DCLK2IRAK1
SCHEMBL6231081 0.80 CFTR (0.47) IRAK4PKMALDH1A1MAPTKMT2A
SCHEMBL6265827 0.79 OPRM1 (0.42) IRAK4PKMALDH1A1MAPTKMT2A
SCHEMBL17487374 0.77 MAPT (0.53) PKMMAPTPOLBKMT2AMEN1
SCHEMBL6275418 0.72 RAB9A (0.47) IRAK4ALDH1A1MAPTPOLBKMT2A
SCHEMBL24900462 0.72 MAPT (0.55) IRAK4PKMALDH1A1MAPTPOLB
SCHEMBL17487406 0.68 MAPT (0.51) PKMALDH1A1MAPTPOLBKMT2A
SCHEMBL9213942 0.68 KDM4E (0.71) IRAK4PKMALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed