SCHEMBL6233688

SCHEMBL6233688

N#Cc1ccccc1S(=O)(=O)N1CCc2cc(Nc3ncnc4cc(C#CN5CCCC5)sc34)ccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.36
ERBB2 P04626 12/20 0.36
PIP4K2A P48426 1/20 0.33
PIP4K2C Q8TBX8 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
HTR6 P50406 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ERBB4 Q15303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271807 0.90 EGFR (0.39) EGFRERBB2PIP4K2APIP4K2CLMNA
SCHEMBL6234112 0.85 ALDH1A1 (0.41) EGFRERBB2PIP4K2APIP4K2CALDH1A1
SCHEMBL6269171 0.84 EGFR (0.41) EGFRERBB2ALDH1A1MAPTERBB4
Formic Acid SCHEMBL6256978 0.83 EGFR (0.46) EGFRERBB2ERBB4
Formic Acid SCHEMBL6256982 0.83 EGFR (0.46) EGFRERBB2ERBB4
SCHEMBL6271804 0.77 EGFR (0.52) EGFRERBB2ERBB4
SCHEMBL6271801 0.77 EGFR (0.52) EGFRERBB2ERBB4
SCHEMBL6269168 0.70 EGFR (0.54) EGFRERBB2ERBB4
SCHEMBL6235814 0.69 EGFR (0.49) EGFRPIP4K2APIP4K2CALDH1A1TDP1
SCHEMBL6239978 0.69 EGFR (0.47) EGFRERBB2ERBB4FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007083-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-27 WO claimed
WO-2005007083-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-27 WO disclosed