SCHEMBL6235814

SCHEMBL6235814

O=S(=O)(Nc1nccs1)c1ccc(Nc2ncnc3cc(C#CN4CCCC4)sc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.49
SCN9A Q15858 1/20 0.43
KDR P35968 2/20 0.43
ALDH1A1 P00352 3/20 0.42
LMNA P02545 3/20 0.42
KDM4E B2RXH2 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
CYP2C9 P11712 1/20 0.42
EDNRA P25101 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA1A P35348 1/20 0.42
PRMT6 Q96LA8 1/20 0.42
ILK Q13418 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
HTT P42858 1/20 0.41
PIP4K2A P48426 1/20 0.41
PIK3R1 P27986 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235809 0.82 EGFR (0.50) EGFRSCN9AKDRALDH1A1LMNA
SCHEMBL6235826 0.82 EGFR (0.50) EGFRSCN9AKDRALDH1A1LMNA
SCHEMBL6234112 0.73 ALDH1A1 (0.41) EGFRALDH1A1PIP4K2APIP4K2CTSHR
SCHEMBL6239978 0.71 EGFR (0.47) EGFR
SCHEMBL6269171 0.71 EGFR (0.41) EGFRKDRALDH1A1MEN1KMT2A
SCHEMBL6236027 0.71 EGFR (0.47) EGFR
Hydrochloric Acid SCHEMBL8812502 0.70 HSD17B10 (0.69) EGFRKDRALDH1A1LMNAKDM4E
SCHEMBL6271807 0.69 EGFR (0.39) EGFRLMNAPIP4K2APIP4K2C
SCHEMBL6233688 0.69 EGFR (0.36) EGFRALDH1A1LMNAKDM4ETDP1
SCHEMBL6252739 0.68 EGFR (0.42) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007083-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-27 WO claimed
WO-2005007083-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-27 WO disclosed