SCHEMBL6234112

SCHEMBL6234112

O=S(=O)(c1cccs1)N1CCc2cc(Nc3ncnc4cc(C#CN5CCCC5)sc34)ccc21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
MKNK1 Q9BUB5 7/20 0.39
TSHR P16473 1/20 0.38
EGFR P00533 5/20 0.38
ERBB2 P04626 4/20 0.38
HPGD P15428 1/20 0.35
PIP4K2A P48426 2/20 0.35
RORC P51449 1/20 0.35
PIP4K2C Q8TBX8 1/20 0.35
FLT1 P17948 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271807 0.86 EGFR (0.39) MKNK1EGFRERBB2PIP4K2APIP4K2C
SCHEMBL6233688 0.85 EGFR (0.36) ALDH1A1EGFRERBB2PIP4K2APIP4K2C
SCHEMBL6269171 0.83 EGFR (0.41) ALDH1A1TSHREGFRERBB2RORC
SCHEMBL6239978 0.82 EGFR (0.47) MKNK1EGFRERBB2FLT1
SCHEMBL6235814 0.73 EGFR (0.49) ALDH1A1TSHREGFRPIP4K2APIP4K2C
SCHEMBL6271801 0.72 EGFR (0.52) EGFRERBB2
SCHEMBL6271804 0.72 EGFR (0.52) EGFRERBB2
SCHEMBL6236350 0.71 FLT1 (0.49) EGFRERBB2FLT1
SCHEMBL6236088 0.70 PIP4K2A (0.40) MKNK1EGFRERBB2PIP4K2A
SCHEMBL6269168 0.70 EGFR (0.54) EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007083-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-27 WO claimed
WO-2005007083-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-27 WO disclosed