SCHEMBL6234327

SCHEMBL6234327

Nc1ccc2nc(CN3CCC(c4ccc(F)cc4)CC3)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.51
MAPT P10636 2/20 0.47
HTR2C P28335 1/20 0.44
ACHE P22303 1/20 0.41
FAAH O00519 1/20 0.40
CYP3A4 P08684 1/20 0.39
DPP4 P27487 1/20 0.39
BACE1 P56817 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
HCRTR1 O43613 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764654 0.88 MCHR1 (0.49) MCHR1FAAHKDM4EMEN1ALDH1A1
SCHEMBL6254675 0.88 MCHR1 (0.53) MCHR1MAPTBACE1
SCHEMBL6233604 0.81 MCHR1 (0.49) MCHR1MAPTHTR2CFAAHCYP3A4
SCHEMBL6230997 0.81 MCHR1 (0.49) MCHR1MAPTHTR2CFAAHCYP3A4
SCHEMBL2921149 0.78 MAOA (0.48) MCHR1MAPTHTR2CACHEFAAH
SCHEMBL6711271 0.78 MAPT (0.57) MCHR1MAPTHTR2CFAAHCYP3A4
SCHEMBL2926351 0.77 ALDH1A1 (0.47) MCHR1MAPTHTR2CACHEFAAH
SCHEMBL6234696 0.76 MAPT (0.41) MCHR1MAPTFAAHKDM4EMEN1
SCHEMBL2918912 0.75 MCHR1 (0.73) MCHR1MAPTHTR2CFAAHKDM4E
SCHEMBL13079397 0.75 MAPT (0.57) MCHR1MAPTHTR2CACHEFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed