SCHEMBL6234788

SCHEMBL6234788

Cn1c(=O)c2ccsc2n(C(=O)O)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 2/20 0.40
ERCC5 P28715 2/20 0.40
FEN1 P39748 2/20 0.40
ERCC4 Q92889 2/20 0.40
ADORA2B P29275 1/20 0.38
HDAC1 Q13547 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KDM1A O60341 1/20 0.34
RCOR1 Q9UKL0 1/20 0.34
CSNK2A1 P68400 2/20 0.34
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6636939 0.72 HTR4 (0.39) ERCC1ERCC5FEN1ERCC4ADORA2B
SCHEMBL7856402 0.72 HTR4 (0.40) ERCC1ERCC5FEN1ERCC4ADORA2B
SCHEMBL13641556 0.65 ADORA1 (0.41) ERCC1ERCC5FEN1ERCC4ADORA2B
SCHEMBL6260462 0.64 ADORA2B (0.40) ERCC1ERCC5FEN1ERCC4ADORA2B
SCHEMBL6513423 0.64 ERCC1 (0.63) ERCC1ERCC5FEN1ERCC4ADORA2B
SCHEMBL11580726 0.61 KMT2A (0.42) MAPTLMNAHSD17B10POLBALDH1A1
SCHEMBL3300277 0.61 ALDH1A1 (0.49) ERCC1FEN1ERCC4LMNAHSD17B10
SCHEMBL4508217 0.61 ALDH1A1 (0.42) MAPTLMNAPOLBALDH1A1EGLN1
SCHEMBL31223899 0.60 LMNA (0.36) ERCC1ERCC5FEN1ERCC4ADORA2B
SCHEMBL20631025 0.60 FEN1 (0.44) ERCC1ERCC5FEN1ERCC4ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed