SCHEMBL62352

SCHEMBL62352

COCNC(=O)C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.42
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
CA2 P00918 4/20 0.36
CA12 O43570 3/20 0.36
CA14 Q9ULX7 1/20 0.36
CA1 P00915 3/20 0.35
CA9 Q16790 2/20 0.35
DGAT1 O75907 1/20 0.34
CA7 P43166 1/20 0.34
DRD2 P14416 4/20 0.34
CTSS P25774 3/20 0.34
CTSK P43235 3/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
EPHX1 P07099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17212001 0.82 CA2 (0.50) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL3275216 0.81 TDP1 (0.36) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL10117371 0.81 TDP1 (0.50) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL17211116 0.79 TDP1 (0.42) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL2089321 0.77 TDP1 (0.41) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL27680256 0.77 TDP1 (0.35) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL4449244 0.75 TDP1 (0.36) TDP1KMT2AMEN1GAACA2
SCHEMBL14152450 0.75 TDP1 (0.36) TDP1KMT2AMEN1GAACA2
SCHEMBL20543014 0.75 TDP1 (0.54) TDP1MAOAMAOBKMT2AMEN1
SCHEMBL19995511 0.75 TDP1 (0.50) TDP1MAOAMAOBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250250244-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H LUNDBECK AS (DK) 2025-08-07 US disclosed
US-12116355-B2 Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia H. LUNDBECK A/S (DK) 2024-10-15 US disclosed
EP-4215512-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H. Lundbeck A/S (DK) 2023-07-26 EP disclosed
EP-3508468-B1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H LUNDBECK AS (DK) 2023-01-18 EP disclosed
US-20220119362-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H. LUNDBECK A/S (DK) 2022-04-21 US disclosed
US-11059798-B2 Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia H. LUNDBECK A/S (DK) 2021-07-13 US disclosed
US-20200131143-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H. LUNDBECK A/S (DK) 2020-04-30 US disclosed
EP-3508468-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H. Lundbeck A/S (DK) 2019-07-10 EP disclosed
US-20190031631-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA H. LUNDBECK A/S (DK) 2019-01-31 US disclosed
US-10118907-B2 Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia H. LUNDBECK A/S (DK) 2018-11-06 US disclosed
US-20120322811-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL-INDANES FOR TREATMENT OF SCHIZOPHRENIA H. LUNDBECK A/S (DK) 2012-12-20 US disclosed
US-8129355-B2 Nuclear receptor-based inducible gene expression system; modulating the expression of a gene in a host cell by introducing into the host cell a gene expression modulation system and activating that system using 5-ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic acid (1-benzoyl-cyclopentyl)-amide INTREXON CORPORATION (US) 2012-03-06 US disclosed
US-8084448-B2 Organic compounds NOVARTIS AG (CH) 2011-12-27 US disclosed
EP-2392561-A1 Alpha-acylaminoketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2011-12-07 EP disclosed
US-20110230464-A1 PURINE DERIVATIVES USEFUL AS P13 KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2011-09-22 US disclosed
US-20090181928-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-07-16 US disclosed
US-20090111183-A1 Ketone Ligands for Modulating the Expression of Exogenous Genes Via An Ecdysone Receptor Complex RHEOGENE, INC. 2009-04-30 US disclosed
US-20080125465-A1 Ketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORPORATION (US) 2008-05-29 US disclosed
US-7375093-B2 Ketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORPORATION (US) 2008-05-20 US disclosed
US-20040049037-A1 Ketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex RHEOGENE, INC. 2004-03-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11059798-B2 Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885
US-20250250244-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885
US-20110230464-A1 PURINE DERIVATIVES USEFUL AS P13 KINASE INHIBITORS PIK3CA, PIK3CD, PI4KA TDP1 350/4885MAOA 2244/4885MAOB 1526/4885
US-20120322811-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL-INDANES FOR TREATMENT OF SCHIZOPHRENIA HTR2C, DRD2, HTR2A TDP1 3408/4885MAOA 280/4885MAOB 232/4885
US-20200131143-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885
US-20220119362-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885
US-20090111183-A1 Ketone Ligands for Modulating the Expression of Exogenous Genes Via An Ecdysone Receptor Complex ESRRB, ESRRA, KDELR1 TDP1 3788/4885MAOA 4519/4885MAOB 4364/4885
US-20090181928-A1 ORGANIC COMPOUNDS PTPRS, PTPRO, PTPRC TDP1 1055/4885MAOA 2048/4885MAOB 1270/4885
US-20190031631-A1 DEUTERATED 1-PIPERAZINO-3-PHENYL INDANES FOR TREATMENT OF SCHIZOPHRENIA HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885
US-20040049037-A1 Ketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex ESRRB, ESRRA, KDELR1 TDP1 3788/4885MAOA 4519/4885MAOB 4364/4885
US-10118907-B2 Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885
US-20080125465-A1 Ketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex ESRRB, ESRRA, KDELR1 TDP1 3788/4885MAOA 4519/4885MAOB 4364/4885
US-12116355-B2 Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia HTR2C, DRD2, HTR2A TDP1 3365/4885MAOA 325/4885MAOB 265/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.