SCHEMBL6236477

SCHEMBL6236477

O=C(CN1CC=C(C2=CC=CCN2)CC1)Nc1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.56
POLB P06746 2/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
KDM4E B2RXH2 3/20 0.52
MAPT P10636 2/20 0.52
LMNA P02545 2/20 0.52
CYP2C19 P33261 4/20 0.49
TSHR P16473 3/20 0.49
CYP2D6 P10635 3/20 0.49
CYP3A4 P08684 3/20 0.49
CYP1A2 P05177 3/20 0.49
USP2 O75604 1/20 0.49
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
LYPLA1 O75608 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
ACHE P22303 1/20 0.43
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237553 0.81 KDM4E (0.48) ALDH1A1KDM4EMAPTLMNACYP2D6
SCHEMBL4004441 0.79 ALDH1A1 (0.65) ALDH1A1POLBL3MBTL1KDM4EMAPT
SCHEMBL6243692 0.78 KDM4E (0.49) ALDH1A1POLBKDM4EMAPTLMNA
SCHEMBL7247601 0.76 KMT2A (0.51) ALDH1A1POLBKDM4EMAPTLMNA
SCHEMBL6243192 0.75 ALDH1A1 (0.56) ALDH1A1KDM4EMAPTCYP2C19TSHR
SCHEMBL6246218 0.74 POLB (0.41) ALDH1A1POLB
SCHEMBL7097274 0.72 ALDH1A1 (0.49) ALDH1A1POLBL3MBTL1KDM4EMAPT
SCHEMBL18657481 0.69 ACHE (0.84) ALDH1A1POLBL3MBTL1KDM4EMAPT
SCHEMBL6245789 0.68 CA1 (0.41) POLBKDM4EMAPTMEN1KMT2A
SCHEMBL8288257 0.66 ALDH1A1 (0.65) ALDH1A1POLBL3MBTL1KDM4ECYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1509213-A2 ACETAMIDES AND BENZAMIDES THAT ARE USEFUL IN TREATING SEXUAL DYSFUNCTION Abbott Laboratories (US) 2005-03-02 EP claimed
WO-2003099266-A2 ACETAMIDES AND BENZAMIDES THAT ARE USEFUL IN TREATING SEXUAL DYSFUNCTION ABBOTT LABORATORIES (US) 2003-12-04 WO claimed