SCHEMBL6236813

SCHEMBL6236813

Cc1ccccc1COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](C)[C@H]2OC(=O)NO)cc1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 16/20 0.59
MMP1 P03956 15/20 0.58
MMP13 P45452 9/20 0.57
S1PR1 P21453 1/20 0.46
S1PR5 Q9H228 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6239853 0.92 ADAM17 (0.51) ADAM17MMP1MMP13
SCHEMBL6241443 0.91 ADAM17 (0.56) ADAM17MMP1MMP13
SCHEMBL6238120 0.91 ADAM17 (0.51) ADAM17MMP1MMP13
SCHEMBL6242757 0.89 MMP1 (0.59) ADAM17MMP1MMP13
SCHEMBL6239672 0.86 ADAM17 (0.44) ADAM17MMP1MMP13
SCHEMBL6238495 0.85 ADAM17 (0.71) ADAM17MMP1MMP13
SCHEMBL6244941 0.84 ADAM17 (0.59) ADAM17MMP1MMP13S1PR1S1PR5
SCHEMBL6238727 0.84 MMP1 (0.54) ADAM17MMP1MMP13
SCHEMBL6237935 0.84 MMP1 (0.52) ADAM17MMP1MMP13
SCHEMBL6238179 0.84 MMP1 (0.54) ADAM17MMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1104412-B1 TACE INHIBITORS PFIZER PROD INC (US) 2005-06-15 EP claimed