SCHEMBL6237018

SCHEMBL6237018

CCNc1nc(C#N)nc(Nc2ccc(C(=O)c3ccccc3)cc2)n1

nearest known ligand 0.74

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.57
CTSK P43235 1/20 0.50
MAPK13 O15264 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
NPC1 O15118 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MMP2 P08253 1/20 0.44
MMP7 P09237 1/20 0.44
MMP10 P09238 1/20 0.44
MMP9 P14780 1/20 0.44
MMP13 P45452 1/20 0.44
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13363711 0.86 TDP1 (0.70) TDP1CTSKADORA2AADORA1
SCHEMBL5257629 0.78 NR1I2 (0.56) TDP1CTSK
SCHEMBL6237210 0.76 TDP1 (0.75) TDP1CTSK
SCHEMBL6239975 0.76 TDP1 (0.56) TDP1CTSKADORA2AADORA1
SCHEMBL6235242 0.74 CTSK (0.76) TDP1CTSKADORA2AADORA1
SCHEMBL5398227 0.73 ALDH1A1 (0.64) MAPK13MAPK12MAPK11MAPK14NPC1
SCHEMBL6236332 0.73 TDP1 (0.66) TDP1CTSK
SCHEMBL6234331 0.72 CTSK (0.68) TDP1CTSKRAB9A
SCHEMBL6240322 0.70 CTSS (0.64) TDP1CTSKADORA2AADORA1
SCHEMBL18510329 0.69 IDH2 (0.52) NPC1CYP1A2CYP2C19RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011703-A1 2-CYANO-1,3,5-TRIAZINE-4,6-DIAMINE DERIVATIVES AKZO NOBEL N.V. (NL) 2005-02-10 WO disclosed
WO-2005011703-A1 2-CYANO-1,3,5-TRIAZINE-4,6-DIAMINE DERIVATIVES AKZO NOBEL N.V. (NL) 2005-02-10 WO disclosed