SCHEMBL6237143

SCHEMBL6237143

Clc1cncc2c1cnn2-c1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.48
GRM1 Q13255 1/20 0.43
CYP2A6 P11509 3/20 0.39
CYP1A2 P05177 2/20 0.38
CYP17A1 P05093 1/20 0.38
GSK3B P49841 1/20 0.37
CYP3A4 P08684 2/20 0.37
METAP2 P50579 1/20 0.36
SCN9A Q15858 1/20 0.36
PIK3CD O00329 1/20 0.35
AOC3 Q16853 1/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HTT P42858 2/20 0.35
CYP2E1 P05181 1/20 0.35
NR3C1 P04150 1/20 0.35
CHRNB2 P17787 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20413782 0.85 ALDH1A1 (0.47) GRM1CYP1A2CYP17A1ALDH1A1NPC1
SCHEMBL15839181 0.84 CYP11B2 (0.48) CYP11B2GRM1CYP2A6CYP1A2CYP17A1
SCHEMBL6276508 0.80 NPC1 (0.46) GRM1ALDH1A1NPC1RAB9AKMT2A
SCHEMBL6278822 0.78 RXFP1 (0.45) CYP11B2CYP1A2CYP17A1GSK3BNPC1
SCHEMBL15839017 0.76 CYP11B2 (0.49) CYP11B2GRM1CYP2A6CYP1A2CYP17A1
SCHEMBL15839068 0.75 CYP11B2 (0.55) CYP11B2GRM1CYP2A6CYP1A2CYP17A1
SCHEMBL6282717 0.73 GSK3B (0.44) CYP11B2GSK3BCYP3A4SCN9A
SCHEMBL6225827 0.73 NPBWR1 (0.39) CYP11B2NPC1RAB9AMAPTPAX8
SCHEMBL15839010 0.72 CYP11B2 (0.56) CYP11B2CYP1A2CYP17A1CYP3A4METAP2
SCHEMBL15839015 0.72 CYP11B2 (0.58) CYP11B2GRM1CYP2A6CYP1A2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1523314-A2 PYRAZOLOPYRIMIDINES AS PROTEIN KINASE INHIBITORS SmithKline Beecham Corporation (US) 2005-04-20 EP disclosed
WO-2004009597-A2 PYRAZOLOPYRIMIDINES AS PROTEIN KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-01-29 WO disclosed