SCHEMBL6237897

SCHEMBL6237897

Cn1c(=O)[nH]c(=O)c2cc(C(=O)OCc3c(Cl)cccc3Cl)sc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.45
ALDH1A1 P00352 6/20 0.45
HSD17B10 Q99714 4/20 0.45
MAPT P10636 4/20 0.45
HPGD P15428 3/20 0.45
TSHR P16473 2/20 0.45
LMNA P02545 2/20 0.45
ESR1 P03372 1/20 0.45
ALOX15 P16050 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
PSMD14 O00487 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
RXFP1 Q9HBX9 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237834 0.84 HSD17B10 (0.45) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6257907 0.84 KDM4E (0.42) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6261894 0.80 KDM4E (0.41) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6254318 0.77 KDM4E (0.43) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6732866 0.77 MAPT (0.44) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6255590 0.75 KDM4E (0.41) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6259014 0.75 HSD17B10 (0.38) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL6256349 0.75 KDM4E (0.36) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL7096960 0.74 MAPT (0.55) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL7100660 0.73 KDM4E (0.36) KDM4EALDH1A1HSD17B10MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed