SCHEMBL6259014

SCHEMBL6259014

Cn1ccc2cc(COC(=O)c3cc4c(=O)[nH]c(=O)n(C)c4s3)ccc21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
HPGD P15428 3/20 0.38
TSHR P16473 2/20 0.38
LMNA P02545 1/20 0.38
ESR1 P03372 1/20 0.38
ALOX15 P16050 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
PSMD14 O00487 1/20 0.37
CHRNA7 P36544 9/20 0.35
KDM4C Q9H3R0 1/20 0.35
TRPV1 Q8NER1 1/20 0.33
HTR2B P41595 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237834 0.81 HSD17B10 (0.45) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6261894 0.80 KDM4E (0.41) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6727703 0.78 MMP13 (0.42) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6257907 0.75 KDM4E (0.42) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6237897 0.75 KDM4E (0.45) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6254318 0.73 KDM4E (0.43) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6255590 0.71 KDM4E (0.41) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6256349 0.71 KDM4E (0.36) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL6257382 0.70 BRD4 (0.48) HSD17B10KDM4EALDH1A1MAPTHPGD
SCHEMBL7100660 0.69 KDM4E (0.36) HSD17B10KDM4EALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed