SCHEMBL6257907

SCHEMBL6257907

Cn1c(=O)[nH]c(=O)c2cc(C(=O)OCc3c(F)c(F)c(F)c(F)c3F)sc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.42
HSD17B10 Q99714 5/20 0.42
ALDH1A1 P00352 5/20 0.42
MAPT P10636 5/20 0.42
HPGD P15428 4/20 0.42
TSHR P16473 2/20 0.42
LMNA P02545 2/20 0.42
ESR1 P03372 2/20 0.42
ALOX15 P16050 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
MMP1 P03956 2/20 0.40
MMP2 P08253 2/20 0.40
MMP9 P14780 2/20 0.40
MMP12 P39900 2/20 0.40
PSMD14 O00487 1/20 0.36
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237897 0.84 KDM4E (0.45) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6237834 0.82 HSD17B10 (0.45) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6261894 0.80 KDM4E (0.41) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6254318 0.80 KDM4E (0.43) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6255590 0.78 KDM4E (0.41) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6256349 0.77 KDM4E (0.36) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL7100660 0.76 KDM4E (0.36) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6259014 0.75 HSD17B10 (0.38) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6254208 0.75 KDM4E (0.43) KDM4EHSD17B10ALDH1A1MAPTHPGD
SCHEMBL6730293 0.74 LMNA (0.49) KDM4EHSD17B10ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed