SCHEMBL623866

SCHEMBL623866

FC(F)(F)Oc1cccc(-c2cnc3sc(N4CC5CNCC5C4)nn23)c1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 8/20 0.48
PIM1 P11309 12/20 0.47
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625741 0.82 PIM1 (0.45) DYRK1APIM1
SCHEMBL623868 0.82 DYRK1A (0.44) DYRK1APIM1KCNH2
SCHEMBL623131 0.82 PIM1 (0.61) DYRK1APIM1KCNH2
SCHEMBL623867 0.82 PIM1 (0.44) PIM1
SCHEMBL623948 0.81 DYRK1A (0.47) DYRK1APIM1KCNH2
SCHEMBL624449 0.80 PIM1 (0.69) DYRK1APIM1KCNH2
SCHEMBL623206 0.80 PIM1 (0.47) DYRK1APIM1KCNH2
SCHEMBL624739 0.80 PIM1 (0.47) DYRK1APIM1KCNH2
SCHEMBL624481 0.79 PIM1 (0.56) DYRK1APIM1KCNH2
SCHEMBL626627 0.78 PIM1 (0.45) DYRK1APIM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed