SCHEMBL624449

SCHEMBL624449

NC1CCCN(c2nn3c(-c4cccc(OC(F)(F)F)c4)cnc3s2)C1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 11/20 0.69
PIM2 Q9P1W9 1/20 0.52
DYRK1A Q13627 5/20 0.47
KCNH2 Q12809 5/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623131 0.94 PIM1 (0.61) PIM1PIM2DYRK1AKCNH2
SCHEMBL625776 0.87 PIM1 (0.55) PIM1PIM2DYRK1AKCNH2
SCHEMBL624450 0.83 PIM1 (0.54) PIM1PIM2
SCHEMBL625254 0.83 PIM3 (0.51) PIM1DYRK1AKCNH2
SCHEMBL623998 0.83 PIM1 (0.51) PIM1PIM2DYRK1AKCNH2
SCHEMBL624481 0.83 PIM1 (0.56) PIM1PIM2DYRK1AKCNH2
SCHEMBL102861 0.82 PIM1 (1.00) PIM1PIM2DYRK1AKCNH2
SCHEMBL140101 0.82 PIM1 (1.00) PIM1PIM2DYRK1AKCNH2
SCHEMBL624016 0.81 PIM1 (0.49) PIM1PIM2KCNH2
SCHEMBL623866 0.80 DYRK1A (0.48) PIM1DYRK1AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed