SCHEMBL6239372

SCHEMBL6239372

CC(C)S(=O)(=O)NC1CCC=C1c1ccc(-c2cccc(NS(C)(=O)=O)c2)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 9/20 0.60
KCNH2 Q12809 5/20 0.57
KIF11 P52732 1/20 0.49
KDM1A O60341 3/20 0.48
TDP2 O95551 2/20 0.43
BRD4 O60885 1/20 0.42
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
AAK1 Q2M2I8 2/20 0.41
FPR2 P25090 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6243992 0.94 GRIA2 (0.58) GRIA2KCNH2KIF11KDM1ATDP2
SCHEMBL6246774 0.85 GRIA2 (0.60) GRIA2KCNH2KDM1ACYP3A4AAK1
SCHEMBL6243805 0.84 GRIA4 (0.44) GRIA2KCNH2KDM1ACYP1A2
SCHEMBL6245808 0.83 CA12 (0.41) GRIA2KCNH2KDM1ACYP1A2
SCHEMBL6239376 0.83 KIF11 (0.47) GRIA2KCNH2KIF11KDM1ATDP2
SCHEMBL6236864 0.80 ADAMTS4 (0.46) GRIA2KCNH2
SCHEMBL6239212 0.79 GRIA2 (0.58) GRIA2KCNH2KDM1ACYP3A4AAK1
SCHEMBL8028031 0.77 GRIA2 (0.65) GRIA2KCNH2KIF11KDM1ATDP2
SCHEMBL6243998 0.77 KIF11 (0.46) GRIA2KCNH2KIF11KDM1ATDP2
SCHEMBL6239207 0.77 GRIA4 (0.44) GRIA2KCNH2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395550-B1 CYCLOALKENYLSULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2005-06-29 EP disclosed
US-20040157817-A1 Cycloalkenylsulfonamide derivatives CANTELL BUDDY EUGENE (US) 2004-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157817-A1 Cycloalkenylsulfonamide derivatives GRIN2B, GRIN2A, GRIN1 GRIA2 7/4885KCNH2 552/4885KIF11 2947/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.