SCHEMBL6239955

SCHEMBL6239955

NC1=CC(N)(CC2CCCO2)NC=C1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 2/20 0.32
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
PKM P14618 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30515668 0.74 ALDH1A1 (0.37) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL6418200 0.70 PDE8B (0.36) ALDH1A1HSD17B10MEN1KMT2ACYP1A2
SCHEMBL3342926 0.65 ALDH1A1 (0.33) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL3341705 0.65 ALDH1A1 (0.33) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL3341702 0.65 ALDH1A1 (0.33) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL3340214 0.65 ALDH1A1 (0.33) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL3342929 0.65 ALDH1A1 (0.33) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL3340212 0.65 ALDH1A1 (0.33) ALDH1A1HPGDTSHRCASP1CASP7
SCHEMBL17437783 0.61 PKM (0.37) ALDH1A1HPGDTSHRPOLBMEN1
SCHEMBL16112324 0.59 TSHR (0.32) ALDH1A1HPGDTSHRPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546129-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS ANTITUMOR AGENT Pharmacia Italia S.p.A. (IT) 2005-06-29 EP disclosed
WO-2004024711-A1 SUBSTITUTED PYRIDINE DERIVATIVES AS ANTITUMOR AGENT PHARMACIA ITALIA S.P.A. (IT) 2004-03-25 WO disclosed