SCHEMBL624037

SCHEMBL624037

CC(C)(C)OC(=O)N1CCC2(CC1)CC(Nc1nn3cc(-c4cccc(C#N)c4)nc3s1)C2

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ADORA2A P29274 1/20 0.39
JAK1 P23458 8/20 0.38
JAK2 O60674 7/20 0.38
MCHR1 Q99705 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
TXK P42681 1/20 0.37
ITK Q08881 1/20 0.37
GPR119 Q8TDV5 2/20 0.37
ROCK2 O75116 1/20 0.37
SCD5 Q86SK9 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623829 0.87 F2RL3 (0.48) JAK2GPR119SCD5SCN9A
SCHEMBL625496 0.86 PIM1 (0.39) HSD17B10IRAK4SCD5
SCHEMBL624036 0.85 FYN (0.46) CYP2D6HSD17B10IRAK4GPR119
SCHEMBL624979 0.82 ADORA2A (0.38) HSD17B10ADORA2AROCK2
SCHEMBL626983 0.82 CETP (0.44) HSD17B10ADORA2AJAK1JAK2GPR119
SCHEMBL625492 0.79 NAMPT (0.39) GPR119
SCHEMBL625408 0.79 MAP4K1 (0.39)
SCHEMBL623873 0.75 IDH1 (0.44) HSD17B10GPR119
SCHEMBL624454 0.75 PIM1 (0.45) GPR119
SCHEMBL625243 0.73 FYN (0.60) JAK2SCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed