SCHEMBL6242523

SCHEMBL6242523

O=c1cnn(-c2ccccc2)c(=O)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNOT7 Q9UIV1 1/20 0.51
HIF1A Q16665 2/20 0.50
DDB1 Q16531 1/20 0.48
CRBN Q96SW2 1/20 0.48
RAB9A P51151 4/20 0.47
ALDH1A1 P00352 4/20 0.47
HTT P42858 3/20 0.47
NPC1 O15118 3/20 0.47
MAPT P10636 2/20 0.47
PAX8 Q06710 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
THRB P10828 2/20 0.47
MITF O75030 1/20 0.47
S1PR4 O95977 1/20 0.47
XBP1 P17861 1/20 0.47
S1PR1 P21453 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
P2RX7 Q99572 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3962079 0.85 NTRK1 (0.51) HIF1AALDH1A1SMN1; SMN2LMNANPSR1
SCHEMBL11784925 0.84 HTR6 (0.43) CNOT7HIF1AALDH1A1HTTLMNA
SCHEMBL30174384 0.81 THRB (0.46) RAB9AALDH1A1HTTNPC1SMN1; SMN2
SCHEMBL7909905 0.81 KMT2A (0.58) RAB9AALDH1A1NPC1SMN1; SMN2LMNA
SCHEMBL30174385 0.81 MEN1 (0.47) RAB9AALDH1A1HTTNPC1MAPT
SCHEMBL10512600 0.81 HIF1A (0.50) HIF1ATHRBP2RX7MEN1NR1I2
SCHEMBL10670742 0.81 P2RX7 (0.43) CNOT7HIF1ARAB9AALDH1A1HTT
SCHEMBL10439328 0.80 MAPK14 (0.45) ALDH1A1HTTMAPTSMN1; SMN2LMNA
SCHEMBL3582300 0.80 TSHR (0.42) DDB1CRBNRAB9ANPC1MAPT
SCHEMBL10439124 0.80 NPC1 (0.55) RAB9AALDH1A1HTTNPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115583919-A Preparation method of 6-oxyalkyl 1,2,4-triazine-3,5 (2H, 4H) -diketone derivative 河北工业大学 2023-01-10 CN claimed
CN-113248454-B Method for preparing 2- [ phenyl ] -1,2, 4-triazine-3, 5(2H,4H) -diketone compound 山东国邦药业有限公司 2021-09-24 CN claimed
CN-113248454-A Method for preparing 2- [ phenyl ] -1,2, 4-triazine-3, 5(2H,4H) -diketone compound 山东国邦药业有限公司 2021-08-13 CN claimed
US-4198407-A Substituted 2-phenyl-1,2,4-triazine-3,5(2H,4H)-diones, and coccidiostatic agents containing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-04-15 US claimed
WO-2026067791-A1 2-PHENYL-1,2,4-TRIAZINE-3,5(2H,4H)-DIONE DERIVATIVES AS THR-BETA AGONIST OR MODULATORS FOR THE TREATMENT OF OBESITY ASCLETIS PHARMA (CHINA) CO., LIMITED (CN) 2026-04-02 WO disclosed
CN-115583919-B Preparation method of 6-oxyalkyl 1,2, 4-triazine-3, 5 (2H, 4H) -diketone derivative 河北工业大学 2024-04-19 CN disclosed
EP-4240730-A1 2-PYRIDONES AS THYROID HORMONE RECEPTOR MODULATORS Aligos Therapeutics, Inc. (US) 2023-09-13 EP disclosed
EP-4240737-A2 BICYCLIC PYRIDAZINONES AS THYROID HORMONE RECEPTOR BETA (TR-BETA) AGONISTS Aligos Therapeutics, Inc. (US) 2023-09-13 EP disclosed
CN-115583919-A Preparation method of 6-oxyalkyl 1,2,4-triazine-3,5 (2H, 4H) -diketone derivative 河北工业大学 2023-01-10 CN disclosed
WO-2022099044-A1 2-PYRIDONES AS THYROID HORMONE RECEPTOR MODULATORS ALIGOS THERAPEUTICS, INC. (US) 2022-05-12 WO disclosed
WO-2022099060-A2 BICYCLIC PYRIDAZINONES AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2022-05-12 WO disclosed
CN-113248454-B Method for preparing 2- [ phenyl ] -1,2, 4-triazine-3, 5(2H,4H) -diketone compound 山东国邦药业有限公司 2021-09-24 CN disclosed
EP-0170316-A2 alpha-Aryl-4-(4,5-dihydro-3,5-dioxo-1,2,4-triazin-2(3H)-yl)benzeneacetonitriles JANSSEN PHARMACEUTICA N.V. (BE) 1986-02-05 EP disclosed
US-4198407-A Substituted 2-phenyl-1,2,4-triazine-3,5(2H,4H)-diones, and coccidiostatic agents containing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-04-15 US disclosed
US-4198407-A Substituted 2-phenyl-1,2,4-triazine-3,5(2H,4H)-diones, and coccidiostatic agents containing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-04-15 US disclosed
US-4198407-A Substituted 2-phenyl-1,2,4-triazine-3,5(2H,4H)-diones, and coccidiostatic agents containing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-04-15 US disclosed
US-3970752-A Coccidiocidal compositions utilizing 1-phenyl-substituted 1,3,5-triazine BAYER AKTIENGESELLSCHAFT (DT) 1976-07-20 US disclosed
US-3948893-A COCCIDIOSIS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-06 US disclosed
US-3912723-A 2-Phenyl-as-triazine-3,5(2H,4H)diones PFIZER 1975-10-14 US disclosed
US-3905971-A 2-Phenyl-as-triazine-3,5(2H,4H)diones PFIZER 1975-09-16 US disclosed