SCHEMBL6242529

SCHEMBL6242529

CCCC(NC(=O)c1ccc(-c2ccccc2)s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.43
CTSS P25774 3/20 0.43
CHRNA7 P36544 5/20 0.36
HTR3E A5X5Y0 4/20 0.36
HTR3B O95264 4/20 0.36
HTR3A P46098 4/20 0.36
HTR3D Q70Z44 4/20 0.36
HTR3C Q8WXA8 4/20 0.36
CTSB P07858 1/20 0.35
P2RY12 Q9H244 1/20 0.35
HPGDS O60760 1/20 0.34
TP53 P04637 1/20 0.34
ACKR3 P25106 4/20 0.34
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
CCR1 P32246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041636 0.92 CTSK (0.47) CTSKCTSSCHRNA7HTR3EHTR3B
SCHEMBL6211260 0.91 CTSK (0.39) CTSKCTSSCHRNA7P2RY12PREP
SCHEMBL4046677 0.89 CTSK (0.34) CTSKCTSSP2RY12
SCHEMBL6274440 0.88 CTSK (0.48) CTSKCTSSP2RY12PREPFAP
SCHEMBL4046318 0.86 CTSK (0.47) CTSKCTSSCHRNA7HTR3EHTR3B
SCHEMBL4048075 0.85 CTSK (0.51) CTSKCTSSCHRNA7HTR3EHTR3B
SCHEMBL4040062 0.84 CTSK (0.40) CTSKCTSSCTSBP2RY12HPGDS
SCHEMBL4045150 0.84 CTSK (0.44) CTSKCTSSP2RY12PREPFAP
SCHEMBL4039142 0.83 CTSK (0.45) CTSKCTSSP2RY12PREPFAP
SCHEMBL6240734 0.83 CTSK (0.39) CTSKCTSSP2RY12PREPFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed